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Dissolution efficiency and bioequivalence study using urine data from healthy volunteers: a comparison between two tablet formulations of cephalexin BJPS
Serra,Cristina Helena dos Reis; Chang,Kyung Hee; Dezani,Thaisa Marinho; Porta,Valentina; Storpirtis,Sílvia.
Tipo: Info:eu-repo/semantics/article Palavras-chave: Tablets/formulations/bioequivalence study; Cephalexin/dissolution efficiency.
Ano: 2015 URL: http://www.scielo.br/scielo.php?script=sci_arttext&pid=S1984-82502015000200383
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Solubility evaluation of didanosine: a comparison between the equilibrium method and intrinsic dissolution for biopharmaceutics classification purposes BJPS
Dezani,André Bersani; Dezani,Thaisa Marinho; Ferreira,Julie Caroline Ferrari; Serra,Cristina Helena dos Reis.
ABSTRACT BCS (Biopharmaceutics Classification System) and BDDCS (Biopharmaceutics Drug Disposition Classification System) were proposed as tools for classifying drugs into four categories. Both systems consider the solubility as an important characteristic for the classification of compounds in drug development and in vivo disposition prediction. Although some results of drug solubility can be found in the literature, the aforementioned characteristic is not entirely clear when considering didanosine (ddI). Based on that, the solubility of ddI was evaluated using equilibrium and intrinsic dissolution methods. For the equilibrium method, excess amount of ddI was added to each media until obtaining a supersaturated solution and the mixture was submitted to...
Tipo: Info:eu-repo/semantics/article Palavras-chave: Didanosine/solubility; Biopharmaceutics Classification System (BCS); Biopharmaceutics Drug Disposition Classification System (BDDCS); Intrinsic dissolution; Equilibrium solubility.
Ano: 2017 URL: http://www.scielo.br/scielo.php?script=sci_arttext&pid=S1984-82502017000200632
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