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Synergistic effect of sertraline and disulfiram against multidrug resistant bacteria as a new alternative to drug repositioning 60
Serafin,Marissa Bolson; Bottega,Angelita; Foletto,Vitória Segabinazzi; Rosa,Taciéli Fagundes da; Rampelotto,Roberta Filipini; Carvalho,Fernanda Aguirre; Hörner,Rosmari.
The repositioning of approved drugs is atopic of interest for the academy and the pharmaceutical industry. The synergistic combination of these drugs can be successful in the treatment of infections caused by resistant bacteria. This study aimed to assess the in vitro synergistic antibacterial activity of sertraline and disulfiram and their interaction with ciprofloxacin and sulfamethoxazole/trimethoprim. We determined the minimum inhibitory concentration, the minimum bactericidal concentration and the fractional inhibitory concentration index. Eighteen bacterial strains were used, being nine American Type Culture Collection reference strains and nine multidrug resistant clinical isolates. Synergy was detected between sertraline and disulfiram against a...
Tipo: Info:eu-repo/semantics/article Palavras-chave: Sertraline; Disulfiram.Antimicrobial activity; Drug synergism; Drug repositioning.
Ano: 2020 URL: http://www.scielo.br/scielo.php?script=sci_arttext&pid=S1984-82502020000100548
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